Josef KA - Search Results

1

Conformationally restrained analogues of pravadoline: nanomolar potent, enantioselective, (aminoalkyl)indole agonists of the cannabinoid receptor.

D'Ambra TE, Estep KG, Bell MR, Eissenstat MA, Josef KA, Ward SJ, Haycock DA, Baizman ER, Casiano FM, Beglin NC, et al. D'Ambra TE, et al. Among authors: josef ka. J Med Chem. 1992 Jan;35(1):124-35. doi: 10.1021/jm00079a016. J Med Chem. 1992. PMID: 1732519

2

Synthesis and structure-activity relationships of 6-heterocyclic-substituted purines as inactivation modifiers of cardiac sodium channels.

Estep KG, Josef KA, Bacon ER, Carabateas PM, Rumney S 4th, Pilling GM, Krafte DS, Volberg WA, Dillon K, Dugrenier N, et al. Estep KG, et al. Among authors: josef ka. J Med Chem. 1995 Jul 7;38(14):2582-95. doi: 10.1021/jm00014a011. J Med Chem. 1995. PMID: 7629798

3

1,3,5-Trialkyl-2,4,6-triiodobenzenes: novel X-ray contrast agents for gastrointestinal imaging.

Estep KG, Josef KA, Bacon ER, Illig CR, Toner JL, Mishra D, Blazak WF, Miller DM, Johnson DK, Allen JM, Spencer A, Wilson SA. Estep KG, et al. Among authors: josef ka. J Med Chem. 2000 May 18;43(10):1940-8. doi: 10.1021/jm990407i. J Med Chem. 2000. PMID: 10821706

4

Pharmacological modulation of human cardiac Na+ channels.

Krafte DS, Davison K, Dugrenier N, Estep K, Josef K, Barchi RL, Kallen RG, Silver PJ, Ezrin AM. Krafte DS, et al. Eur J Pharmacol. 1994 Feb 15;266(3):245-54. doi: 10.1016/0922-4106(94)90133-3. Eur J Pharmacol. 1994. PMID: 8174607

5

1,2-Benzothiazine 1,1-dioxide P(2)-P(3) peptide mimetic aldehyde calpain I inhibitors.

Wells GJ, Tao M, Josef KA, Bihovsky R. Wells GJ, et al. Among authors: josef ka. J Med Chem. 2001 Oct 11;44(21):3488-503. doi: 10.1021/jm010178b. J Med Chem. 2001. PMID: 11585453

6

4,5-dihydropyridazin-3-one derivatives as histamine H₃ receptor inverse agonists.

Hudkins RL, Aimone LD, Dandu RR, Dunn D, Gruner JA, Huang Z, Josef KA, Lyons JA, Mathiasen JR, Tao M, Zulli AL, Raddatz R. Hudkins RL, et al. Among authors: josef ka. Bioorg Med Chem Lett. 2012 Jan 1;22(1):194-8. doi: 10.1016/j.bmcl.2011.11.037. Epub 2011 Nov 16. Bioorg Med Chem Lett. 2012. PMID: 22142542

7

Synthesis and biological activity of a series of potent fluoromethyl ketone inhibitors of recombinant human calpain I.

Chatterjee S, Ator MA, Bozyczko-Coyne D, Josef K, Wells G, Tripathy R, Iqbal M, Bihovsky R, Senadhi SE, Mallya S, O'Kane TM, McKenna BA, Siman R, Mallamo JP. Chatterjee S, et al. J Med Chem. 1997 Nov 7;40(23):3820-8. doi: 10.1021/jm970197e. J Med Chem. 1997. PMID: 9371247

8

Identification of pyridazin-3-one derivatives as potent, selective histamine H₃ receptor inverse agonists with robust wake activity.

Hudkins RL, Aimone LD, Bailey TR, Bendesky RJ, Dandu RR, Dunn D, Gruner JA, Josef KA, Lin YG, Lyons J, Marcy VR, Mathiasen JR, Sundar BG, Tao M, Zulli AL, Raddatz R, Bacon ER. Hudkins RL, et al. Among authors: josef ka. Bioorg Med Chem Lett. 2011 Sep 15;21(18):5493-7. doi: 10.1016/j.bmcl.2011.06.108. Epub 2011 Jun 30. Bioorg Med Chem Lett. 2011. PMID: 21782432

9

Synthesis of constrained benzocinnolinone analogues of CEP-26401 (irdabisant) as potent, selective histamine H3 receptor inverse agonists.

Josef KA, Aimone LD, Lyons J, Raddatz R, Hudkins RL. Josef KA, et al. Bioorg Med Chem Lett. 2012 Jun 15;22(12):4198-202. doi: 10.1016/j.bmcl.2012.04.001. Epub 2012 Apr 26. Bioorg Med Chem Lett. 2012. PMID: 22617490

10

D-amino acid containing, high-affinity inhibitors of recombinant human calpain I.

Chatterjee S, Gu ZQ, Dunn D, Tao M, Josef K, Tripathy R, Bihovsky R, Senadhi SE, O'Kane TM, McKenna BA, Mallya S, Ator MA, Bozyczko-Coyne D, Siman R, Mallamo JP. Chatterjee S, et al. J Med Chem. 1998 Jul 16;41(15):2663-6. doi: 10.1021/jm980035y. J Med Chem. 1998. PMID: 9667954 No abstract available.

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