Bruns RF - Search Results

1

Structure-activity relationships of a series of benzothiophene-derived NPY Y1 antagonists: optimization of the C-2 side chain.

Britton TC, Spinazze PG, Hipskind PA, Zimmerman DM, Zarrinmayeh H, Schober DA, Gehlert DR, Bruns RF. Britton TC, et al. Among authors: bruns rf. Bioorg Med Chem Lett. 1999 Feb 8;9(3):475-80. doi: 10.1016/s0960-894x(99)00019-0. Bioorg Med Chem Lett. 1999. PMID: 10091705

2

Synthesis and evaluation of a series of novel 2-[(4-chlorophenoxy)methyl]benzimidazoles as selective neuropeptide Y Y1 receptor antagonists.

Zarrinmayeh H, Nunes AM, Ornstein PL, Zimmerman DM, Arnold MB, Schober DA, Gackenheimer SL, Bruns RF, Hipskind PA, Britton TC, Cantrell BE, Gehlert DR. Zarrinmayeh H, et al. Among authors: bruns rf. J Med Chem. 1998 Jul 16;41(15):2709-19. doi: 10.1021/jm9706630. J Med Chem. 1998. PMID: 9667962

3

Structure-activity relationships of a series of 1-substituted-4-methylbenzimidazole neuropeptide Y-1 receptor antagonists.

Zimmerman DM, Cantrell BE, Smith EC, Nixon JA, Bruns RF, Gitter B, Hipskind PA, Ornstein PL, Zarrinmayeh H, Britton TC, Schober DA, Gehlert DR. Zimmerman DM, et al. Among authors: bruns rf. Bioorg Med Chem Lett. 1998 Mar 3;8(5):473-6. doi: 10.1016/s0960-894x(98)00048-1. Bioorg Med Chem Lett. 1998. PMID: 9871601

4

Structure-activity relationship of a series of diaminoalkyl substituted benzimidazole as neuropeptide Y Y1 receptor antagonists.

Zarrinmayeh H, Zimmerman DM, Cantrell BE, Schober DA, Bruns RF, Gackenheimer SL, Ornstein PL, Hipskind PA, Britton TC, Gehlert DR. Zarrinmayeh H, et al. Among authors: bruns rf. Bioorg Med Chem Lett. 1999 Mar 8;9(5):647-52. doi: 10.1016/s0960-894x(99)00082-7. Bioorg Med Chem Lett. 1999. PMID: 10201822

5

3-Aryl-1,2-diacetamidopropane derivatives as novel and potent NK-1 receptor antagonists.

Hipskind PA, Howbert JJ, Bruns RF, Cho SS, Crowell TA, Foreman MM, Gehlert DR, Iyengar S, Johnson KW, Krushinski JH, Li DL, Lobb KL, Mason NR, Muehl BS, Nixon JA, Phebus LA, Regoli D, Simmons RM, Threlkeld PG, Waters DC, Gitter BD. Hipskind PA, et al. Among authors: bruns rf. J Med Chem. 1996 Feb 2;39(3):736-48. doi: 10.1021/jm950616c. J Med Chem. 1996. PMID: 8576917

6

Potent and selective 1,2,3-trisubstituted indole NPY Y-1 antagonists.

Hipskind PA, Lobb KL, Nixon JA, Britton TC, Bruns RF, Catlow J, Dieckman-McGinty DK, Gackenheimer SL, Gitter BD, Iyengar S, Schober DA, Simmons RM, Swanson S, Zarrinmayeh H, Zimmerman DM, Gehlert DR. Hipskind PA, et al. Among authors: bruns rf. J Med Chem. 1997 Nov 7;40(23):3712-4. doi: 10.1021/jm970512x. J Med Chem. 1997. PMID: 9371234 No abstract available.

7

The neuropeptide Y Y1 antagonist, 1229U91, a potent agonist for the human pancreatic polypeptide-preferring (NPY Y4) receptor.

Schober DA, Van Abbema AM, Smiley DL, Bruns RF, Gehlert DR. Schober DA, et al. Among authors: bruns rf. Peptides. 1998;19(3):537-42. doi: 10.1016/s0196-9781(97)00455-5. Peptides. 1998. PMID: 9533642

8

An Allosteric Potentiator of the Dopamine D1 Receptor Increases Locomotor Activity in Human D1 Knock-In Mice without Causing Stereotypy or Tachyphylaxis.

Svensson KA, Heinz BA, Schaus JM, Beck JP, Hao J, Krushinski JH, Reinhard MR, Cohen MP, Hellman SL, Getman BG, Wang X, Menezes MM, Maren DL, Falcone JF, Anderson WH, Wright RA, Morin SM, Knopp KL, Adams BL, Rogovoy B, Okun I, Suter TM, Statnick MA, Gehlert DR, Nelson DL, Lucaites VL, Emkey R, DeLapp NW, Wiernicki TR, Cramer JW, Yang CR, Bruns RF. Svensson KA, et al. Among authors: bruns rf. J Pharmacol Exp Ther. 2017 Jan;360(1):117-128. doi: 10.1124/jpet.116.236372. Epub 2016 Nov 3. J Pharmacol Exp Ther. 2017. PMID: 27811173 Free PMC article.

9

[1,2,4]Triazolo[4,3-a]quinoxalin-4-amines: a new class of A1 receptor selective adenosine antagonists.

Trivedi BK, Bruns RF. Trivedi BK, et al. Among authors: bruns rf. J Med Chem. 1988 May;31(5):1011-4. doi: 10.1021/jm00400a021. J Med Chem. 1988. PMID: 3361571

10

C2,N6-disubstituted adenosines: synthesis and structure-activity relationships.

Trivedi BK, Bruns RF. Trivedi BK, et al. Among authors: bruns rf. J Med Chem. 1989 Aug;32(8):1667-73. doi: 10.1021/jm00128a002. J Med Chem. 1989. PMID: 2754691

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