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A series of C-terminal amino alcohol dipeptide A beta inhibitors.
Bioorg Med Chem Lett. 2002 Nov 4;12(21):3051-3. doi: 10.1016/s0960-894x(02)00684-4.
Bioorg Med Chem Lett. 2002.
PMID: 12372499
Discovery of a novel [3.2.1] benzo fused bicyclic sulfonamide-pyrazoles as potent, selective and efficacious γ-secretase inhibitors.
Ye XM, Konradi AW, Sun M, Yuan S, Aubele DL, Dappen M, Dressen D, Garofalo AW, Jagodzinski JJ, Latimer L, Probst GD, Sham HL, Wone D, Xu YZ, Ness D, Brigham E, Kwong GT, Willtis C, Tonn G, Goldbach E, Quinn KP, Zhang HH, Sauer JM, Bova M, Basi GS.
Ye XM, et al.
Bioorg Med Chem Lett. 2013 Feb 15;23(4):996-1000. doi: 10.1016/j.bmcl.2012.12.039. Epub 2012 Dec 21.
Bioorg Med Chem Lett. 2013.
PMID: 23312944
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Preparation and optimization of a series of 3-carboxamido-5-phenacylaminopyrazole bradykinin B1 receptor antagonists.
Dressen D, Garofalo AW, Hawkinson J, Hom D, Jagodzinski J, Marugg JL, Neitzel ML, Pleiss MA, Szoke B, Tung JS, Wone DW, Wu J, Zhang H.
Dressen D, et al. Among authors: wone dw.
J Med Chem. 2007 Oct 18;50(21):5161-7. doi: 10.1021/jm051292n. Epub 2007 Sep 19.
J Med Chem. 2007.
PMID: 17880055
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Design and synthesis of cell potent BACE-1 inhibitors: structure-activity relationship of P1' substituents.
Sealy JM, Truong AP, Tso L, Probst GD, Aquino J, Hom RK, Jagodzinska BM, Dressen D, Wone DW, Brogley L, John V, Tung JS, Pleiss MA, Tucker JA, Konradi AW, Dappen MS, Toth G, Pan H, Ruslim L, Miller J, Bova MP, Sinha S, Quinn KP, Sauer JM.
Sealy JM, et al. Among authors: wone dw.
Bioorg Med Chem Lett. 2009 Nov 15;19(22):6386-91. doi: 10.1016/j.bmcl.2009.09.061. Epub 2009 Sep 19.
Bioorg Med Chem Lett. 2009.
PMID: 19811916
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Optimizing phenylethylphosphonamidates for the inhibition of prostate-specific membrane antigen.
Wone DW, Rowley JA, Garofalo AW, Berkman CE.
Wone DW, et al.
Bioorg Med Chem. 2006 Jan 1;14(1):67-76. doi: 10.1016/j.bmc.2005.07.056. Epub 2005 Sep 9.
Bioorg Med Chem. 2006.
PMID: 16154750
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Design of an orally efficacious hydroxyethylamine (HEA) BACE-1 inhibitor in a preclinical animal model.
Truong AP, Tóth G, Probst GD, Sealy JM, Bowers S, Wone DW, Dressen D, Hom RK, Konradi AW, Sham HL, Wu J, Peterson BT, Ruslim L, Bova MP, Kholodenko D, Motter RN, Bard F, Santiago P, Ni H, Chian D, Soriano F, Cole T, Brigham EF, Wong K, Zmolek W, Goldbach E, Samant B, Chen L, Zhang H, Nakamura DF, Quinn KP, Yednock TA, Sauer JM.
Truong AP, et al. Among authors: wone dw.
Bioorg Med Chem Lett. 2010 Nov 1;20(21):6231-6. doi: 10.1016/j.bmcl.2010.08.102. Epub 2010 Aug 24.
Bioorg Med Chem Lett. 2010.
PMID: 20833041
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Development of a novel β-secretase binding assay using the AlphaScreen platform.
Ren Z, Tam D, Xu YZ, Wone D, Yuan S, Sham HL, Cheung H, Regnstrom K, Chen X, Rudolph D, Jobling MF, Artis DR, Bova MP.
Ren Z, et al.
J Biomol Screen. 2013 Jul;18(6):695-704. doi: 10.1177/1087057113482138. Epub 2013 Mar 29.
J Biomol Screen. 2013.
PMID: 23543430
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