Jeyakumar M - Search Results

1

Dual-mode fluorophore-doped nickel nitrilotriacetic acid-modified silica nanoparticles combine histidine-tagged protein purification with site-specific fluorophore labeling.

Kim SH, Jeyakumar M, Katzenellenbogen JA. Kim SH, et al. Among authors: jeyakumar m. J Am Chem Soc. 2007 Oct 31;129(43):13254-64. doi: 10.1021/ja074443f. Epub 2007 Oct 2. J Am Chem Soc. 2007. PMID: 17910454 Free PMC article.

2

Exploration of dimensions of estrogen potency: parsing ligand binding and coactivator binding affinities.

Jeyakumar M, Carlson KE, Gunther JR, Katzenellenbogen JA. Jeyakumar M, et al. J Biol Chem. 2011 Apr 15;286(15):12971-82. doi: 10.1074/jbc.M110.205112. Epub 2011 Feb 14. J Biol Chem. 2011. PMID: 21321128 Free PMC article.

3

Quantification of ligand-regulated nuclear receptor corepressor and coactivator binding, key interactions determining ligand potency and efficacy for the thyroid hormone receptor.

Jeyakumar M, Webb P, Baxter JD, Scanlan TS, Katzenellenbogen JA. Jeyakumar M, et al. Biochemistry. 2008 Jul 15;47(28):7465-76. doi: 10.1021/bi800393u. Epub 2008 Jun 18. Biochemistry. 2008. PMID: 18558711 Free PMC article.

4

A dual-acceptor time-resolved Föster resonance energy transfer assay for simultaneous determination of thyroid hormone regulation of corepressor and coactivator binding to the thyroid hormone receptor: Mimicking the cellular context of thyroid hormone action.

Jeyakumar M, Katzenellenbogen JA. Jeyakumar M, et al. Anal Biochem. 2009 Mar 1;386(1):73-8. doi: 10.1016/j.ab.2008.11.039. Epub 2008 Dec 7. Anal Biochem. 2009. PMID: 19111515 Free PMC article.

5

Diarylpropionitrile (DPN) enantiomers: synthesis and evaluation of estrogen receptor β-selective ligands.

Carroll VM, Jeyakumar M, Carlson KE, Katzenellenbogen JA. Carroll VM, et al. Among authors: jeyakumar m. J Med Chem. 2012 Jan 12;55(1):528-37. doi: 10.1021/jm201436k. Epub 2011 Dec 14. J Med Chem. 2012. PMID: 22122563 Free PMC article.

6

Synthesis and biological evaluation of two agents for imaging estrogen receptor β by positron emission tomography: challenges in PET imaging of a low abundance target.

Lee JH, Peters O, Lehmann L, Dence CS, Sharp TL, Carlson KE, Zhou D, Jeyakumar M, Welch MJ, Katzenellenbogen JA. Lee JH, et al. Among authors: jeyakumar m. Nucl Med Biol. 2012 Nov;39(8):1105-16. doi: 10.1016/j.nucmedbio.2012.05.011. Epub 2012 Jun 30. Nucl Med Biol. 2012. PMID: 22749433 Free PMC article.

7

Mechanisms enforcing the estrogen receptor β selectivity of botanical estrogens.

Jiang Y, Gong P, Madak-Erdogan Z, Martin T, Jeyakumar M, Carlson K, Khan I, Smillie TJ, Chittiboyina AG, Rotte SC, Helferich WG, Katzenellenbogen JA, Katzenellenbogen BS. Jiang Y, et al. Among authors: jeyakumar m. FASEB J. 2013 Nov;27(11):4406-18. doi: 10.1096/fj.13-234617. Epub 2013 Jul 23. FASEB J. 2013. PMID: 23882126 Free PMC article.

8

Raloxifene and ICI182,780 increase estrogen receptor-alpha association with a nuclear compartment via overlapping sets of hydrophobic amino acids in activation function 2 helix 12.

Lupien M, Jeyakumar M, Hébert E, Hilmi K, Cotnoir-White D, Loch C, Auger A, Dayan G, Pinard GA, Wurtz JM, Moras D, Katzenellenbogen J, Mader S. Lupien M, et al. Among authors: jeyakumar m. Mol Endocrinol. 2007 Apr;21(4):797-816. doi: 10.1210/me.2006-0074. Epub 2007 Feb 13. Mol Endocrinol. 2007. PMID: 17299137

9

Small-animal PET of steroid hormone receptors predicts tumor response to endocrine therapy using a preclinical model of breast cancer.

Fowler AM, Chan SR, Sharp TL, Fettig NM, Zhou D, Dence CS, Carlson KE, Jeyakumar M, Katzenellenbogen JA, Schreiber RD, Welch MJ. Fowler AM, et al. Among authors: jeyakumar m. J Nucl Med. 2012 Jul;53(7):1119-26. doi: 10.2967/jnumed.112.103465. Epub 2012 Jun 5. J Nucl Med. 2012. PMID: 22669982 Free PMC article.

10

Phosphorylation of thyroid hormone receptor-associated nuclear receptor corepressor holocomplex by the DNA-dependent protein kinase enhances its histone deacetylase activity.

Jeyakumar M, Liu XF, Erdjument-Bromage H, Tempst P, Bagchi MK. Jeyakumar M, et al. J Biol Chem. 2007 Mar 30;282(13):9312-9322. doi: 10.1074/jbc.M609009200. Epub 2007 Jan 22. J Biol Chem. 2007. PMID: 17242407 Free article.

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