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Novel ATP competitive MK2 inhibitors with potent biochemical and cell-based activity throughout the series.
Oubrie A, Kaptein A, de Zwart E, Hoogenboom N, Goorden R, van de Kar B, van Hoek M, de Kimpe V, van der Heijden R, Borsboom J, Kazemier B, de Roos J, Scheffers M, Lommerse J, Schultz-Fademrecht C, Barf T. Oubrie A, et al. Among authors: van de kar b, van hoek m, van der heijden r. Bioorg Med Chem Lett. 2012 Jan 1;22(1):613-8. doi: 10.1016/j.bmcl.2011.10.071. Epub 2011 Nov 3. Bioorg Med Chem Lett. 2012. PMID: 22119462
Structure-based lead identification of ATP-competitive MK2 inhibitors.
Barf T, Kaptein A, de Wilde S, van der Heijden R, van Someren R, Demont D, Schultz-Fademrecht C, Versteegh J, van Zeeland M, Seegers N, Kazemier B, van de Kar B, van Hoek M, de Roos J, Klop H, Smeets R, Hofstra C, Hornberg J, Oubrie A. Barf T, et al. Among authors: van someren r, van de kar b, van zeeland m, van hoek m, van der heijden r. Bioorg Med Chem Lett. 2011 Jun 15;21(12):3818-22. doi: 10.1016/j.bmcl.2011.04.018. Epub 2011 Apr 16. Bioorg Med Chem Lett. 2011. PMID: 21565500
Post-traumatic and OA-related lesions in the knee at baseline and 2 years after traumatic meniscal injury: Secondary analysis of a randomized controlled trial.
van der Graaff SJA, Oei EHG, Reijman M, Steenbekkers L, van Middelkoop M, van der Heijden RA, Meuffels DE; STARR Study Group. van der Graaff SJA, et al. Among authors: van der heijden ra. Osteoarthritis Cartilage. 2024 Apr 2:S1063-4584(24)01132-4. doi: 10.1016/j.joca.2024.03.116. Online ahead of print. Osteoarthritis Cartilage. 2024. PMID: 38574801 Free article.
The ISMRM Open Science Initiative for Perfusion Imaging (OSIPI): Results from the OSIPI-Dynamic Contrast-Enhanced challenge.
Shalom ES, Kim H, van der Heijden RA, Ahmed Z, Patel R, Hormuth DA 2nd, DiCarlo JC, Yankeelov TE, Sisco NJ, Dortch RD, Stokes AM, Inglese M, Grech-Sollars M, Toschi N, Sahoo P, Singh A, Verma SK, Rathore DK, Kazerouni AS, Partridge SC, LoCastro E, Paudyal R, Wolansky IA, Shukla-Dave A, Schouten P, Gurney-Champion OJ, Jiřík R, Macíček O, Bartoš M, Vitouš J, Das AB, Kim SG, Bokacheva L, Mikheev A, Rusinek H, Berks M, Hubbard Cristinacce PL, Little RA, Cheung S, O'Connor JPB, Parker GJM, Moloney B, LaViolette PS, Bobholz S, Duenweg S, Virostko J, Laue HO, Sung K, Nabavizadeh A, Saligheh Rad H, Hu LS, Sourbron S, Bell LC, Fathi Kazerooni A. Shalom ES, et al. Among authors: van der heijden ra. Magn Reson Med. 2024 May;91(5):1803-1821. doi: 10.1002/mrm.29909. Epub 2023 Dec 19. Magn Reson Med. 2024. PMID: 38115695
Perfusion Imaging of the Musculoskeletal System.
Griffith JF, Yip SWY, van der Heijden RA, Valenzuela RF, Yeung DKW. Griffith JF, et al. Among authors: van der heijden ra. Magn Reson Imaging Clin N Am. 2024 Feb;32(1):181-206. doi: 10.1016/j.mric.2023.07.004. Epub 2023 Oct 8. Magn Reson Imaging Clin N Am. 2024. PMID: 38007280 Review.
Up-and-coming Radiotracers for Imaging Pain Generators.
van der Heijden RA, Biswal S. van der Heijden RA, et al. Semin Musculoskelet Radiol. 2023 Dec;27(6):661-675. doi: 10.1055/s-0043-1775745. Epub 2023 Nov 7. Semin Musculoskelet Radiol. 2023. PMID: 37935213 Free PMC article.
Advanced Magnetic Resonance Imaging and Molecular Imaging of the Painful Knee.
Mostert JM, Dur NBJ, Li X, Ellermann JM, Hemke R, Hales L, Mazzoli V, Kogan F, Griffith JF, Oei EHG, van der Heijden RA. Mostert JM, et al. Among authors: van der heijden ra. Semin Musculoskelet Radiol. 2023 Dec;27(6):618-631. doi: 10.1055/s-0043-1775741. Epub 2023 Nov 7. Semin Musculoskelet Radiol. 2023. PMID: 37935208 Free PMC article. Review.
A community-endorsed open-source lexicon for contrast agent-based perfusion MRI: A consensus guidelines report from the ISMRM Open Science Initiative for Perfusion Imaging (OSIPI).
Dickie BR, Ahmed Z, Arvidsson J, Bell LC, Buckley DL, Debus C, Fedorov A, Floca R, Gutmann I, van der Heijden RA, van Houdt PJ, Sourbron S, Thrippleton MJ, Quarles C, Kompan IN; on behalf of The Perfusion Study Group of the ISMRM. Dickie BR, et al. Among authors: van der heijden ra. Magn Reson Med. 2024 May;91(5):1761-1773. doi: 10.1002/mrm.29840. Epub 2023 Oct 13. Magn Reson Med. 2024. PMID: 37831600
171 results