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A Potent and Selective AMPK Activator That Inhibits de Novo Lipogenesis.
ACS Med Chem Lett. 2010 Aug 30;1(9):478-82. doi: 10.1021/ml100143q. eCollection 2010 Dec 9.
ACS Med Chem Lett. 2010.
PMID: 24900234
Free PMC article.
Synthesis and characterization of a novel liver-targeted prodrug of cytosine-1-beta-D-arabinofuranoside monophosphate for the treatment of hepatocellular carcinoma.
Boyer SH, Sun Z, Jiang H, Esterbrook J, Gómez-Galeno JE, Craigo W, Reddy KR, Ugarkar BG, MacKenna DA, Erion MD.
Boyer SH, et al.
J Med Chem. 2006 Dec 28;49(26):7711-20. doi: 10.1021/jm0607449.
J Med Chem. 2006.
PMID: 17181153
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Pradefovir: a prodrug that targets adefovir to the liver for the treatment of hepatitis B.
Reddy KR, Matelich MC, Ugarkar BG, Gómez-Galeno JE, DaRe J, Ollis K, Sun Z, Craigo W, Colby TJ, Fujitaki JM, Boyer SH, van Poelje PD, Erion MD.
Reddy KR, et al.
J Med Chem. 2008 Feb 14;51(3):666-76. doi: 10.1021/jm7012216. Epub 2008 Jan 4.
J Med Chem. 2008.
PMID: 18173234
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Design of highly active analogues of the pyrrolo[1,2-a]benzimidazole antitumor agents.
Craigo WA, LeSueur BW, Skibo EB.
Craigo WA, et al.
J Med Chem. 1999 Aug 26;42(17):3324-33. doi: 10.1021/jm990029h.
J Med Chem. 1999.
PMID: 10464019
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Pyrimidoquinazoline-based antitumor agents. Design of topoisomerase II to DNA cross-linkers with activity against protein kinases.
Skibo EB, Huang X, Martinez R, Lemus RH, Craigo WA, Dorr RT.
Skibo EB, et al. Among authors: craigo wa.
J Med Chem. 2002 Dec 5;45(25):5543-55. doi: 10.1021/jm020285l.
J Med Chem. 2002.
PMID: 12459022
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