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Preparation and biological evaluation of conformationally constrained BACE1 inhibitors.
Bioorg Med Chem. 2015 Jul 1;23(13):3260-8. doi: 10.1016/j.bmc.2015.04.062. Epub 2015 May 6.
Bioorg Med Chem. 2015.
PMID: 26001341
Preparation and biological evaluation of BACE1 inhibitors: Leveraging trans-cyclopropyl moieties as ligand efficient conformational constraints.
Winneroski LL, Erickson JA, Green SJ, Lopez JE, Stout SL, Porter WJ, Timm DE, Audia JE, Barberis M, Beck JP, Boggs LN, Borders AR, Boyer RD, Brier RA, Hembre EJ, Hendle J, Garcia-Losada P, Minguez JM, Mathes BM, May PC, Monk SA, Rankovic Z, Shi Y, Watson BM, Yang Z, Mergott DJ.
Winneroski LL, et al. Among authors: garcia losada p.
Bioorg Med Chem. 2020 Jan 1;28(1):115194. doi: 10.1016/j.bmc.2019.115194. Epub 2019 Nov 15.
Bioorg Med Chem. 2020.
PMID: 31786008
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Discovery and Early Clinical Development of LY3202626, a Low-Dose, CNS-Penetrant BACE Inhibitor.
McKinzie DL, Winneroski LL, Green SJ, Hembre EJ, Erickson JA, Willis BA, Monk SA, Aluise CD, Baker TK, Lopez JE, Hendle J, Beck JP, Brier RA, Boggs LN, Borders AR, Cocke PJ, Garcia-Losada P, Lowe SL, Mathes BM, May PC, Porter WJ, Stout SL, Timm DE, Watson BM, Yang Z, Mergott DJ.
McKinzie DL, et al. Among authors: garcia losada p.
J Med Chem. 2021 Jun 24;64(12):8076-8100. doi: 10.1021/acs.jmedchem.1c00489. Epub 2021 Jun 3.
J Med Chem. 2021.
PMID: 34081466
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Development of a selective androgen receptor modulator for transdermal use in hypogonadal patients.
Krishnan V, Patel NJ, Mackrell JG, Sweetana SA, Bullock H, Ma YL, Waterhouse TH, Yaden BC, Henck J, Zeng QQ, Gavardinas K, Jadhav P, Saeed A, Garcia-Losada P, Robins DA, Benson CT.
Krishnan V, et al. Among authors: garcia losada p.
Andrology. 2018 May;6(3):455-464. doi: 10.1111/andr.12479. Epub 2018 Mar 12.
Andrology. 2018.
PMID: 29527831
Free article.
Clinical Trial.
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Accelerated and Scalable C(sp3)-H Amination via Decatungstate Photocatalysis Using a Flow Photoreactor Equipped with High-Intensity LEDs.
Wan T, Wen Z, Laudadio G, Capaldo L, Lammers R, Rincón JA, García-Losada P, Mateos C, Frederick MO, Broersma R, Noël T.
Wan T, et al. Among authors: garcia losada p.
ACS Cent Sci. 2022 Jan 26;8(1):51-56. doi: 10.1021/acscentsci.1c01109. Epub 2021 Dec 16.
ACS Cent Sci. 2022.
PMID: 35106372
Free PMC article.
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The Merger of Benzophenone HAT Photocatalysis and Silyl Radical-Induced XAT Enables Both Nickel-Catalyzed Cross-Electrophile Coupling and 1,2-Dicarbofunctionalization of Olefins.
Luridiana A, Mazzarella D, Capaldo L, Rincón JA, García-Losada P, Mateos C, Frederick MO, Nuño M, Jan Buma W, Noël T.
Luridiana A, et al. Among authors: garcia losada p.
ACS Catal. 2022 Sep 16;12(18):11216-11225. doi: 10.1021/acscatal.2c03805. Epub 2022 Sep 1.
ACS Catal. 2022.
PMID: 36158902
Free PMC article.
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Decatungstate-Mediated C(sp3 )-H Heteroarylation via Radical-Polar Crossover in Batch and Flow.
Wan T, Capaldo L, Laudadio G, Nyuchev AV, Rincón JA, García-Losada P, Mateos C, Frederick MO, Nuño M, Noël T.
Wan T, et al. Among authors: garcia losada p.
Angew Chem Int Ed Engl. 2021 Aug 9;60(33):17893-17897. doi: 10.1002/anie.202104682. Epub 2021 Jul 9.
Angew Chem Int Ed Engl. 2021.
PMID: 34060204
Free PMC article.
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Electrochemical Nickel-Catalyzed C(sp3)-C(sp3) Cross-Coupling of Alkyl Halides with Alkyl Tosylates.
Ibrahim MYS, Cumming GR, Gonzalez de Vega R, Garcia-Losada P, de Frutos O, Kappe CO, Cantillo D.
Ibrahim MYS, et al. Among authors: garcia losada p.
J Am Chem Soc. 2023 Aug 9;145(31):17023-17028. doi: 10.1021/jacs.3c07313. Epub 2023 Jul 26.
J Am Chem Soc. 2023.
PMID: 37494617
Free PMC article.
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