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Synthesis of 1'-C-cyano pyrimidine nucleosides and characterization as HCV polymerase inhibitors.
Nucleosides Nucleotides Nucleic Acids. 2015;34(11):763-85. doi: 10.1080/15257770.2015.1075550. Epub 2015 Sep 23.
Nucleosides Nucleotides Nucleic Acids. 2015.
PMID: 26398773
A palladium-catalyzed alkylation/direct arylation synthesis of nitrogen-containing heterocycles.
Blaszykowski C, Aktoudianakis E, Alberico D, Bressy C, Hulcoop DG, Jafarpour F, Joushaghani A, Laleu B, Lautens M.
Blaszykowski C, et al. Among authors: aktoudianakis e.
J Org Chem. 2008 Mar 7;73(5):1888-97. doi: 10.1021/jo702052b. Epub 2008 Feb 9.
J Org Chem. 2008.
PMID: 18260672
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Preparation of annulated nitrogen-containing heterocycles via a one-pot palladium-catalyzed alkylation/direct arylation sequence.
Blaszykowski C, Aktoudianakis E, Bressy C, Alberico D, Lautens M.
Blaszykowski C, et al. Among authors: aktoudianakis e.
Org Lett. 2006 May 11;8(10):2043-5. doi: 10.1021/ol060447y.
Org Lett. 2006.
PMID: 16671777
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Discovery of Hepatitis B Virus Surface Antigen Suppressor GS-8873.
Kato D, Choy RW, Canales E, Dick RA, Lake AD, Shapiro ND, Chin E, Li J, Zhang JR, Wu Q, Saito RD, Metobo S, Aktoudianakis E, Schroeder SD, Yang ZY, Glatt DM, Balsitis S, Gamelin L, Yu M, Cheng G, Delaney WE 4th, Link JO.
Kato D, et al. Among authors: aktoudianakis e.
ACS Med Chem Lett. 2024 Mar 22;15(4):546-554. doi: 10.1021/acsmedchemlett.4c00037. eCollection 2024 Apr 11.
ACS Med Chem Lett. 2024.
PMID: 38628802
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