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Page 1
Novel bicyclo[3.1.0]hexane analogs as antagonists of metabotropic glutamate 2/3 receptors for the treatment of depression.
Dressman BA, Tromiczak EG, Chappell MD, Tripp AE, Quimby SJ, Vetman T, Fivush AM, Matt J, Jaramillo C, Li R, Khilevich A, Blanco MJ, Smith SC, Carpintero M, de Diego JE, Barberis M, García-Cerrada S, Soriano JF, Schkeryantz JM, Witkin JM, Wafford KA, Seidel W, Britton T, Overshiner CD, Li X, Wang XS, Heinz BA, Catlow JT, Swanson S, Bedwell D, Ornstein PL, Mitch CH. Dressman BA, et al. Among authors: barberis m. Bioorg Med Chem Lett. 2016 Dec 1;26(23):5663-5668. doi: 10.1016/j.bmcl.2016.10.067. Epub 2016 Oct 25. Bioorg Med Chem Lett. 2016. PMID: 27836401
Imidazolyl benzimidazoles and imidazo[4,5-b]pyridines as potent p38alpha MAP kinase inhibitors with excellent in vivo antiinflammatory properties.
Mader M, de Dios A, Shih C, Bonjouklian R, Li T, White W, López de Uralde B, Sánchez-Martinez C, del Prado M, Jaramillo C, de Diego E, Martín Cabrejas LM, Dominguez C, Montero C, Shepherd T, Dally R, Toth JE, Chatterjee A, Pleite S, Blanco-Urgoiti J, Perez L, Barberis M, Lorite MJ, Jambrina E, Nevill CR Jr, Lee PA, Schultz RC, Wolos JA, Li LC, Campbell RM, Anderson BD. Mader M, et al. Among authors: barberis m. Bioorg Med Chem Lett. 2008 Jan 1;18(1):179-83. doi: 10.1016/j.bmcl.2007.10.106. Epub 2007 Nov 1. Bioorg Med Chem Lett. 2008. PMID: 18039577
Discovery of (1S,2R,3S,4S,5R,6R)-2-Amino-3-[(3,4-difluorophenyl)sulfanylmethyl]-4-hydroxy-bicyclo[3.1.0]hexane-2,6-dicarboxylic Acid Hydrochloride (LY3020371·HCl): A Potent, Metabotropic Glutamate 2/3 Receptor Antagonist with Antidepressant-Like Activity.
Chappell MD, Li R, Smith SC, Dressman BA, Tromiczak EG, Tripp AE, Blanco MJ, Vetman T, Quimby SJ, Matt J, Britton TC, Fivush AM, Schkeryantz JM, Mayhugh D, Erickson JA, Bures MG, Jaramillo C, Carpintero M, Diego JE, Barberis M, Garcia-Cerrada S, Soriano JF, Antonysamy S, Atwell S, MacEwan I, Condon B, Sougias C, Wang J, Zhang A, Conners K, Groshong C, Wasserman SR, Koss JW, Witkin JM, Li X, Overshiner C, Wafford KA, Seidel W, Wang XS, Heinz BA, Swanson S, Catlow JT, Bedwell DW, Monn JA, Mitch CH, Ornstein PL. Chappell MD, et al. Among authors: barberis m. J Med Chem. 2016 Dec 22;59(24):10974-10993. doi: 10.1021/acs.jmedchem.6b01119. Epub 2016 Dec 6. J Med Chem. 2016. PMID: 28002967
Preparation and biological evaluation of BACE1 inhibitors: Leveraging trans-cyclopropyl moieties as ligand efficient conformational constraints.
Winneroski LL, Erickson JA, Green SJ, Lopez JE, Stout SL, Porter WJ, Timm DE, Audia JE, Barberis M, Beck JP, Boggs LN, Borders AR, Boyer RD, Brier RA, Hembre EJ, Hendle J, Garcia-Losada P, Minguez JM, Mathes BM, May PC, Monk SA, Rankovic Z, Shi Y, Watson BM, Yang Z, Mergott DJ. Winneroski LL, et al. Among authors: barberis m. Bioorg Med Chem. 2020 Jan 1;28(1):115194. doi: 10.1016/j.bmc.2019.115194. Epub 2019 Nov 15. Bioorg Med Chem. 2020. PMID: 31786008
Synthesis of Enantiopure Unnatural Amino Acids by Metallaphotoredox Catalysis.
Faraggi TM, Rouget-Virbel C, Rincón JA, Barberis M, Mateos C, García-Cerrada S, Agejas J, de Frutos O, MacMillan DWC. Faraggi TM, et al. Among authors: barberis m. Org Process Res Dev. 2021 Aug 20;25(8):1966-1973. doi: 10.1021/acs.oprd.1c00208. Epub 2021 Jul 26. Org Process Res Dev. 2021. PMID: 35663840 Free PMC article.
Discovery of potent small-molecule inhibitors of lipoprotein(a) formation.
Diaz N, Perez C, Escribano AM, Sanz G, Priego J, Lafuente C, Barberis M, Calle L, Espinosa JF, Priest BT, Zhang HY, Nosie AK, Haas JV, Cannady E, Borel A, Schultze AE, Sauder JM, Hendle J, Weichert K, Nicholls SJ, Michael LF. Diaz N, et al. Among authors: barberis m. Nature. 2024 May;629(8013):945-950. doi: 10.1038/s41586-024-07387-z. Epub 2024 May 8. Nature. 2024. PMID: 38720069 Free PMC article.
Clinical actionability of BRCA2 alterations in uterine leiomyosarcoma: a molecular tumor board case report and a cBioPortal comprehensive analysis.
Boscolo Bielo L, Repetto M, Crimini E, Belli C, Setola E, Parma G, Fusco N, Barberis M, Guerini Rocco E, Marra A, Colombo N, Curigliano G. Boscolo Bielo L, et al. Among authors: barberis m. Oncologist. 2024 May 8:oyae082. doi: 10.1093/oncolo/oyae082. Online ahead of print. Oncologist. 2024. PMID: 38716772 Free article.
Knowledge, attitudes and perceptions of Latin American healthcare workers relating to antibiotic stewardship and antibiotic use: a cross-sectional multi-country study.
Fabre V, Cosgrove SE, Lessa FC, Patel TS, Reyes-Morales G, Aleman WR, Alvarez AA, Aquiles B, Arauz AB, Arguello F, Barberis MF, Barcan L, Bernachea MP, Bernan ML, Buitrago C, Del Carmen Bangher M, Castañeda X, Colque AM, Canton A, Contreras R, Correa S, Campero GC, Espinola L, Esquivel C, Ezcurra C, Falleroni LA, Fernandez J, Ferrari S, Frassone N, Cruz CG, Garzón MI, Quintero CHG, Gonzalez JA, Guaymas L, Guerrero-Toapanta F, Lambert S, Laplume D, Lazarte PR, Lemir CG, Lopez A, Lopez IL, Maldonado H, Martinez G, Maurizi DM, Melgar M, Mesplet F, Pertuz CM, Moreno C, Moya GL, Nuccetelli Y, Núñez G, Osuna C, Palacio B, Pellice F, Raffo C, Choto FR, Ricoy G, Rodriguez V, Romero F, Romero JJ, Russo ME, Sadino G, Sandoval N, Silva MG, Urueña AM, Reyes LV, Videla H, Valle M, Perez SVA, Vergara-Samur H, Villamandos S, Villarreal O, Viteri A, Warley E, Quiros RE. Fabre V, et al. Among authors: barberis mf. Antimicrob Resist Infect Control. 2024 Apr 26;13(1):47. doi: 10.1186/s13756-024-01400-w. Antimicrob Resist Infect Control. 2024. PMID: 38664757 Free PMC article.
392 results