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Discovery of (1S,2R,3S,4S,5R,6R)-2-Amino-3-[(3,4-difluorophenyl)sulfanylmethyl]-4-hydroxy-bicyclo[3.1.0]hexane-2,6-dicarboxylic Acid Hydrochloride (LY3020371·HCl): A Potent, Metabotropic Glutamate 2/3 Receptor Antagonist with Antidepressant-Like Activity.
J Med Chem. 2016 Dec 22;59(24):10974-10993. doi: 10.1021/acs.jmedchem.6b01119. Epub 2016 Dec 6.
J Med Chem. 2016.
PMID: 28002967
Rapid-access, high-throughput synchrotron crystallography for drug discovery.
Wasserman SR, Koss JW, Sojitra ST, Morisco LL, Burley SK.
Wasserman SR, et al. Among authors: koss jw.
Trends Pharmacol Sci. 2012 May;33(5):261-7. doi: 10.1016/j.tips.2012.03.009. Epub 2012 Apr 18.
Trends Pharmacol Sci. 2012.
PMID: 22521107
Review.
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Automated electron microscopy for evaluating two-dimensional crystallization of membrane proteins.
Hu M, Vink M, Kim C, Derr K, Koss J, D'Amico K, Cheng A, Pulokas J, Ubarretxena-Belandia I, Stokes D.
Hu M, et al.
J Struct Biol. 2010 Jul;171(1):102-10. doi: 10.1016/j.jsb.2010.02.018. Epub 2010 Mar 1.
J Struct Biol. 2010.
PMID: 20197095
Free PMC article.
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