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IMI European Lead Factory - democratizing access to high-throughput screening.
Nat Rev Drug Discov. 2022 Apr;21(4):245-246. doi: 10.1038/d41573-021-00196-3.
Nat Rev Drug Discov. 2022.
PMID: 34907316
No abstract available.
The European Lead Factory: An updated HTS compound library for innovative drug discovery.
van Vlijmen H, Ortholand JY, Li VM, de Vlieger JSB.
van Vlijmen H, et al. Among authors: ortholand jy.
Drug Discov Today. 2021 Oct;26(10):2406-2413. doi: 10.1016/j.drudis.2021.04.019. Epub 2021 Apr 20.
Drug Discov Today. 2021.
PMID: 33892142
Free article.
Review.
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Corrigendum to "The European Lead Factory: An updated HTS compound library for innovative drug discovery" [Drug Discov. Today 26(10) (2021) 2406-2413].
van Vlijmen H, Ortholand JY, Li VM, de Vlieger JSB.
van Vlijmen H, et al. Among authors: ortholand jy.
Drug Discov Today. 2023 Aug;28(8):103257. doi: 10.1016/j.drudis.2022.04.005. Epub 2022 Apr 7.
Drug Discov Today. 2023.
PMID: 35398021
No abstract available.
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Exploring new targets and chemical space with affinity selection-mass spectrometry.
Prudent R, Annis DA, Dandliker PJ, Ortholand JY, Roche D.
Prudent R, et al. Among authors: ortholand jy.
Nat Rev Chem. 2021 Jan;5(1):62-71. doi: 10.1038/s41570-020-00229-2. Epub 2020 Oct 21.
Nat Rev Chem. 2021.
PMID: 37118102
Review.
Item in Clipboard
The European Lead Factory: Results from a decade of collaborative, public-private, drug discovery programs.
van Vlijmen H, Pannifer AD, Cochrane P, Basting D, Li VM, Engkvist O, Ortholand JY, Wagener M, Duffy J, Finsinger D, Davis J, van Helden SP, de Vlieger JSB; European Lead Factory Consortium.
van Vlijmen H, et al. Among authors: ortholand jy.
Drug Discov Today. 2024 Mar;29(3):103886. doi: 10.1016/j.drudis.2024.103886. Epub 2024 Jan 18.
Drug Discov Today. 2024.
PMID: 38244673
Free article.
Review.
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Rhodium(III)-catalyzed allylic C-H bond amination. Synthesis of cyclic amines from ω-unsaturated N-sulfonylamines.
Cochet T, Bellosta V, Roche D, Ortholand JY, Greiner A, Cossy J.
Cochet T, et al. Among authors: ortholand jy.
Chem Commun (Camb). 2012 Nov 11;48(87):10745-7. doi: 10.1039/c2cc36067e.
Chem Commun (Camb). 2012.
PMID: 23023187
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Isolation and kinetic properties of acetohydroxy acid isomeroreductase from spinach (Spinacia oleracea) chloroplasts overexpressed in Escherichia coli.
Dumas R, Job D, Ortholand JY, Emeric G, Greiner A, Douce R.
Dumas R, et al. Among authors: ortholand jy.
Biochem J. 1992 Dec 15;288 ( Pt 3)(Pt 3):865-74. doi: 10.1042/bj2880865.
Biochem J. 1992.
PMID: 1472001
Free PMC article.
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Natural products and combinatorial chemistry: back to the future.
Ortholand JY, Ganesan A.
Ortholand JY, et al.
Curr Opin Chem Biol. 2004 Jun;8(3):271-80. doi: 10.1016/j.cbpa.2004.04.011.
Curr Opin Chem Biol. 2004.
PMID: 15183325
Review.
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