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Identification of SARS-CoV-2 Mpro inhibitors containing P1' 4-fluorobenzothiazole moiety highly active against SARS-CoV-2.
Higashi-Kuwata N, Tsuji K, Hayashi H, Bulut H, Kiso M, Imai M, Ogata-Aoki H, Ishii T, Kobayakawa T, Nakano K, Takamune N, Kishimoto N, Hattori SI, Das D, Uemura Y, Shimizu Y, Aoki M, Hasegawa K, Suzuki S, Nishiyama A, Saruwatari J, Shimizu Y, Sukenaga Y, Takamatsu Y, Tsuchiya K, Maeda K, Yoshimura K, Iida S, Ozono S, Suzuki T, Okamura T, Misumi S, Kawaoka Y, Tamamura H, Mitsuya H. Higashi-Kuwata N, et al. Among authors: okamura t. Nat Commun. 2023 Feb 25;14(1):1076. doi: 10.1038/s41467-023-36729-0. Nat Commun. 2023. PMID: 36841831 Free PMC article.
Novel murine model of congenital diabetes: The insulin hyposecretion mouse.
Nakano K, Yanobu-Takanashi R, Takahashi Y, Sasaki H, Shimizu Y, Okamura T, Sasaki N. Nakano K, et al. Among authors: okamura t. J Diabetes Investig. 2019 Mar;10(2):227-237. doi: 10.1111/jdi.12895. Epub 2018 Aug 17. J Diabetes Investig. 2019. PMID: 29987871 Free PMC article.
Acute Respiratory Infection in Human Dipeptidyl Peptidase 4-Transgenic Mice Infected with Middle East Respiratory Syndrome Coronavirus.
Iwata-Yoshikawa N, Okamura T, Shimizu Y, Kotani O, Sato H, Sekimukai H, Fukushi S, Suzuki T, Sato Y, Takeda M, Tashiro M, Hasegawa H, Nagata N. Iwata-Yoshikawa N, et al. Among authors: okamura t. J Virol. 2019 Mar 5;93(6):e01818-18. doi: 10.1128/JVI.01818-18. Print 2019 Mar 15. J Virol. 2019. PMID: 30626685 Free PMC article.
GRL-0920, an Indole Chloropyridinyl Ester, Completely Blocks SARS-CoV-2 Infection.
Hattori SI, Higshi-Kuwata N, Raghavaiah J, Das D, Bulut H, Davis DA, Takamatsu Y, Matsuda K, Takamune N, Kishimoto N, Okamura T, Misumi S, Yarchoan R, Maeda K, Ghosh AK, Mitsuya H. Hattori SI, et al. Among authors: okamura t. mBio. 2020 Aug 20;11(4):e01833-20. doi: 10.1128/mBio.01833-20. mBio. 2020. PMID: 32820005 Free PMC article.
Fibroblasts as a source of self-antigens for central immune tolerance.
Nitta T, Tsutsumi M, Nitta S, Muro R, Suzuki EC, Nakano K, Tomofuji Y, Sawa S, Okamura T, Penninger JM, Takayanagi H. Nitta T, et al. Among authors: okamura t. Nat Immunol. 2020 Oct;21(10):1172-1180. doi: 10.1038/s41590-020-0756-8. Epub 2020 Aug 24. Nat Immunol. 2020. PMID: 32839611
2,838 results