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Small molecule drug metabolite synthesis and identification: why, when and how?
Drug Discov Today. 2024 May;29(5):103943. doi: 10.1016/j.drudis.2024.103943. Epub 2024 Mar 5.
Drug Discov Today. 2024.
PMID: 38452922
Free article.
Review.
Open Source Antibiotics: Simple Diarylimidazoles Are Potent against Methicillin-Resistant Staphylococcus aureus.
Klug DM, Tse EG, Silva DG, Cao Y, Charman SA, Chauhan J, Crighton E, Dichiara M, Drake C, Drewry D, da Silva Emery F, Ferrins L, Graves L, Hopkins E, Kresina TAC, Lorente-Macías Á, Perry B, Phipps R, Quiroga B, Quotadamo A, Sabatino GN, Sama A, Schätzlein A, Simpson QJ, Steele J, Shanu-Wilson J, Sjö P, Stapleton P, Swain CJ, Vaideanu A, Xie H, Zuercher W, Todd MH.
Klug DM, et al. Among authors: shanu wilson j.
ACS Infect Dis. 2023 Dec 8;9(12):2423-2435. doi: 10.1021/acsinfecdis.3c00286. Epub 2023 Nov 22.
ACS Infect Dis. 2023.
PMID: 37991879
Free PMC article.
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Biotransformation: Impact and Application of Metabolism in Drug Discovery.
Shanu-Wilson J, Evans L, Wrigley S, Steele J, Atherton J, Boer J.
Shanu-Wilson J, et al.
ACS Med Chem Lett. 2020 Aug 28;11(11):2087-2107. doi: 10.1021/acsmedchemlett.0c00202. eCollection 2020 Nov 12.
ACS Med Chem Lett. 2020.
PMID: 33214818
Free PMC article.
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