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Discovery and SAR Study of Boronic Acid-Based Selective PDE3B Inhibitors from a Novel DNA-Encoded Library.
J Med Chem. 2024 Feb 8;67(3):2049-2065. doi: 10.1021/acs.jmedchem.3c01562. Epub 2024 Jan 29.
J Med Chem. 2024.
PMID: 38284310
Discovery of a Novel 2,6-Disubstituted Glucosamine Series of Potent and Selective Hexokinase 2 Inhibitors.
Lin H, Zeng J, Xie R, Schulz MJ, Tedesco R, Qu J, Erhard KF, Mack JF, Raha K, Rendina AR, Szewczuk LM, Kratz PM, Jurewicz AJ, Cecconie T, Martens S, McDevitt PJ, Martin JD, Chen SB, Jiang Y, Nickels L, Schwartz BJ, Smallwood A, Zhao B, Campobasso N, Qian Y, Briand J, Rominger CM, Oleykowski C, Hardwicke MA, Luengo JI.
Lin H, et al. Among authors: cecconie t.
ACS Med Chem Lett. 2015 Dec 28;7(3):217-22. doi: 10.1021/acsmedchemlett.5b00214. eCollection 2016 Mar 10.
ACS Med Chem Lett. 2015.
PMID: 26985301
Free PMC article.
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Targeting the Regulatory Site of ER Aminopeptidase 1 Leads to the Discovery of a Natural Product Modulator of Antigen Presentation.
Liddle J, Hutchinson JP, Kitchen S, Rowland P, Neu M, Cecconie T, Holmes DS, Jones E, Korczynska J, Koumantou D, Lea JD, Nickels L, Pemberton M, Phillipou A, Schneck JL, Sheehan H, Tinworth CP, Uings I, Wojno-Picon J, Young RJ, Stratikos E.
Liddle J, et al. Among authors: cecconie t.
J Med Chem. 2020 Mar 26;63(6):3348-3358. doi: 10.1021/acs.jmedchem.9b02123. Epub 2020 Mar 9.
J Med Chem. 2020.
PMID: 32109056
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Discovery of Proline-Based p300/CBP Inhibitors Using DNA-Encoded Library Technology in Combination with High-Throughput Screening.
Tian X, Suarez D, Thomson D, Li W, King EA, LaFrance L, Boehm J, Barton L, Di Marco C, Martyr C, Thalji R, Medina J, Knight S, Heerding D, Gao E, Nartey E, Cecconie T, Nixon C, Zhang G, Berrodin TJ, Phelps C, Patel A, Bai X, Lind K, Prabhu N, Messer J, Zhu Z, Shewchuk L, Reid R, Graves AP, McHugh C, Mangatt B.
Tian X, et al. Among authors: cecconie t.
J Med Chem. 2022 Nov 10;65(21):14391-14408. doi: 10.1021/acs.jmedchem.2c00670. Epub 2022 Oct 27.
J Med Chem. 2022.
PMID: 36302181
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Biochemical and functional characterization of the p.A165T missense variant of mitochondrial amidoxime-reducing component 1.
Hou W, Watson C, Cecconie T, Bolaki MN, Brady JJ, Lu Q, Gatto GJ Jr, Day TA.
Hou W, et al. Among authors: cecconie t.
J Biol Chem. 2024 May 7:107353. doi: 10.1016/j.jbc.2024.107353. Online ahead of print.
J Biol Chem. 2024.
PMID: 38723751
Free article.
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Theory and practice of ubiquitous quantitative chemical analysis using conventional computer optical disk drives.
Potyrailo RA, Morris WG, Leach AM, Hassib L, Krishnan K, Surman C, Wroczynski R, Boyette S, Xiao C, Shrikhande P, Agree A, Cecconie T.
Potyrailo RA, et al. Among authors: cecconie t.
Appl Opt. 2007 Oct 1;46(28):7007-17. doi: 10.1364/ao.46.007007.
Appl Opt. 2007.
PMID: 17906730
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