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Series of (([1,1'-Biphenyl]-2-yl)methyl)sulfinylalkyl Alicyclic Amines as Novel and High Affinity Atypical Dopamine Transporter Inhibitors with Reduced hERG Activity.
ACS Pharmacol Transl Sci. 2024 Jan 5;7(2):515-532. doi: 10.1021/acsptsci.3c00322. eCollection 2024 Feb 9.
ACS Pharmacol Transl Sci. 2024.
PMID: 38357284
Modifications to 1-(4-(2-Bis(4-fluorophenyl)methyl)sulfinyl)alkyl Alicyclic Amines That Improve Metabolic Stability and Retain an Atypical DAT Inhibitor Profile.
Okorom AV, Camacho-Hernandez GA, Salomon K, Lee KH, Ku TC, Cao J, Won SJ, Friedman J, Lam J, Paule J, Rais R, Klein B, Xi ZX, Shi L, Loland CJ, Newman AH.
Okorom AV, et al.
J Med Chem. 2024 Jan 11;67(1):709-727. doi: 10.1021/acs.jmedchem.3c02037. Epub 2023 Dec 20.
J Med Chem. 2024.
PMID: 38117239
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Dynamic extracellular vestibule of human SERT: Unveiling druggable potential with high-affinity allosteric inhibitors.
Salomon K, Abramyan AM, Plenge P, Wang L, Bundgaard C, Bang-Andersen B, Loland CJ, Shi L.
Salomon K, et al.
Proc Natl Acad Sci U S A. 2023 Oct 10;120(41):e2304089120. doi: 10.1073/pnas.2304089120. Epub 2023 Oct 4.
Proc Natl Acad Sci U S A. 2023.
PMID: 37792512
Free PMC article.
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The antidepressant drug vilazodone is an allosteric inhibitor of the serotonin transporter.
Plenge P, Yang D, Salomon K, Laursen L, Kalenderoglou IE, Newman AH, Gouaux E, Coleman JA, Loland CJ.
Plenge P, et al.
Nat Commun. 2021 Aug 20;12(1):5063. doi: 10.1038/s41467-021-25363-3.
Nat Commun. 2021.
PMID: 34417466
Free PMC article.
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