Triarylpyrazoles with basic side chains: development of pyrazole-based estrogen receptor antagonists.
Stauffer SR, Huang YR, Aron ZD, Coletta CJ, Sun J, Katzenellenbogen BS, Katzenellenbogen JA.
Stauffer SR, et al. Among authors: sun j.
Bioorg Med Chem. 2001 Jan;9(1):151-61. doi: 10.1016/s0968-0896(00)00226-1.
Bioorg Med Chem. 2001.
PMID: 11197335
.: Mortenson, D. S.: Stauffer, S. R.; Aron, Z. D.: Katzenellenbogen, J. A. Chem. Biol. 1999, 6, 205). Subsequent work has shown that some analogues in this series are very selective for the ERalpha subtype in terms of binding affinity and agonist potency (Stauffer, S. R.: …
.: Mortenson, D. S.: Stauffer, S. R.; Aron, Z. D.: Katzenellenbogen, J. A. Chem. Biol. 1999, 6, 205). Subsequent work has shown that …