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(R)-3,3,3-Trifluoro-2-hydroxy-2-methylpropionamides are orally active inhibitors of pyruvate dehydrogenase kinase.
J Med Chem. 1999 Jul 29;42(15):2741-6. doi: 10.1021/jm9902584.
J Med Chem. 1999.
PMID: 10425084
No abstract available.
Triterpene and diterpene inhibitors of pyruvate dehydrogenase kinase (PDK).
Aicher TD, Damon RE, Koletar J, Vinluan CC, Brand LJ, Gao J, Shetty SS, Kaplan EL, Mann WR.
Aicher TD, et al. Among authors: vinluan cc.
Bioorg Med Chem Lett. 1999 Aug 2;9(15):2223-8. doi: 10.1016/s0960-894x(99)00380-7.
Bioorg Med Chem Lett. 1999.
PMID: 10465550
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Secondary amides of (R)-3,3,3-trifluoro-2-hydroxy-2-methylpropionic acid as inhibitors of pyruvate dehydrogenase kinase.
Aicher TD, Anderson RC, Gao J, Shetty SS, Coppola GM, Stanton JL, Knorr DC, Sperbeck DM, Brand LJ, Vinluan CC, Kaplan EL, Dragland CJ, Tomaselli HC, Islam A, Lozito RJ, Liu X, Maniara WM, Fillers WS, DelGrande D, Walter RE, Mann WR.
Aicher TD, et al. Among authors: vinluan cc.
J Med Chem. 2000 Jan 27;43(2):236-49. doi: 10.1021/jm990358+.
J Med Chem. 2000.
PMID: 10649979
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Anilides of (R)-trifluoro-2-hydroxy-2-methylpropionic acid as inhibitors of pyruvate dehydrogenase kinase.
Bebernitz GR, Aicher TD, Stanton JL, Gao J, Shetty SS, Knorr DC, Strohschein RJ, Tan J, Brand LJ, Liu C, Wang WH, Vinluan CC, Kaplan EL, Dragland CJ, DelGrande D, Islam A, Lozito RJ, Liu X, Maniara WM, Mann WR.
Bebernitz GR, et al. Among authors: vinluan cc.
J Med Chem. 2000 Jun 1;43(11):2248-57. doi: 10.1021/jm0000923.
J Med Chem. 2000.
PMID: 10841803
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Diverse mechanisms of inhibition of pyruvate dehydrogenase kinase by structurally distinct inhibitors.
Mann WR, Dragland CJ, Vinluan CC, Vedananda TR, Bell PA, Aicher TD.
Mann WR, et al. Among authors: vinluan cc.
Biochim Biophys Acta. 2000 Jul 14;1480(1-2):283-92. doi: 10.1016/s0167-4838(00)00079-0.
Biochim Biophys Acta. 2000.
PMID: 11004568
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Heterologously expressed inner lipoyl domain of dihydrolipoyl acetyltransferase inhibits ATP-dependent inactivation of pyruvate dehydrogenase complex. Identification of important amino acid residues.
Jackson JC, Vinluan CC, Dragland CJ, Sundararajan V, Yan B, Gounarides JS, Nirmala NR, Topiol S, Ramage P, Blume JE, Aicher TD, Bell PA, Mann WR.
Jackson JC, et al. Among authors: vinluan cc.
Biochem J. 1998 Sep 15;334 ( Pt 3)(Pt 3):703-11. doi: 10.1042/bj3340703.
Biochem J. 1998.
PMID: 9729480
Free PMC article.
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