Reversal of subtype-selectivity and function by the introduction of a para-benzamidyl substituent to N-cyclopropylmethyl nornepenthone.
Kong L, Ning K, Liu X, Lu J, Chen B, Ye R, Li Z, Jiang S, Tang S, Chai JR, Fang Y, Lan Y, Mai X, Xie Q, Liu J, Shao L, Fu W, Wang Y, Li W.
Kong L, et al. Among authors: chai jr.
Eur J Med Chem. 2023 Oct 5;258:115589. doi: 10.1016/j.ejmech.2023.115589. Epub 2023 Jun 28.
Eur J Med Chem. 2023.
PMID: 37413884